SCHEMBL28294439

SCHEMBL28294439

O=C(NCC1(CO)CCC1)c1cc[c]cn1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.49
P2RX7 Q99572 2/20 0.41
CNR1 P21554 3/20 0.37
JAK2 O60674 2/20 0.34
JAK1 P23458 2/20 0.34
TYK2 P29597 2/20 0.34
JAK3 P52333 2/20 0.34
CACNA1H O95180 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21379657 0.73 CNR2 (0.49) CNR2P2RX7
SCHEMBL749356 0.72 CNR1 (0.42) CNR1
SCHEMBL28292579 0.72 CNR2 (0.50) CNR2P2RX7CNR1
SCHEMBL28294346 0.69 CNR2 (0.41) CNR2
SCHEMBL30333324 0.68 CNR2 (0.52) CNR2P2RX7CNR1JAK2JAK1
SCHEMBL422451 0.67 CNR1 (0.38) CNR1
SCHEMBL752887 0.66 CHRM2 (0.44) CNR1
SCHEMBL753368 0.66 POLB (0.56) CNR1
SCHEMBL15776856 0.66 CNR2 (1.00) CNR2CNR1
SCHEMBL13162890 0.66 P2RX7 (0.56) CNR2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed