SCHEMBL28292579

SCHEMBL28292579

NC(=O)Oc1ccc(C(=O)NCC2(CO)CCC2)nc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.50
P2RX7 Q99572 2/20 0.40
MAOB P27338 1/20 0.35
SCN9A Q15858 1/20 0.35
CNR1 P21554 1/20 0.35
BACE1 P56817 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28940931 0.87 CNR2 (0.40) CNR2MAOBSCN9ABACE1
SCHEMBL28292566 0.79 MAOB (0.49) MAOBSCN9ACNR1
SCHEMBL21379657 0.76 CNR2 (0.49) CNR2P2RX7
SCHEMBL28292577 0.73 CCNC (0.48) CNR2MAOBSCN9A
SCHEMBL28940932 0.72 CNR2 (0.49) CNR2MAOBSCN9A
SCHEMBL28940985 0.72 SCN9A (0.44) MAOBSCN9A
SCHEMBL28292586 0.72 SCN9A (0.44) MAOBSCN9A
SCHEMBL28294439 0.72 CNR2 (0.49) CNR2P2RX7CNR1
SCHEMBL28284688 0.71 CCNC (0.43) CNR1HRH3
SCHEMBL28294317 0.71 SCN9A (0.45) MAOBSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed