SCHEMBL28294520

SCHEMBL28294520

CCc1ccn(C)n1.NCc1ccc(-c2nc(Cn3cccn3)cs2)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 15/20 0.45
KLK1 P06870 13/20 0.44
PLG P00747 1/20 0.40
PRSS1 P07477 1/20 0.40
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28296211 0.88 KLKB1 (0.43) KLKB1KLK1PLGPRSS1NPC1
SCHEMBL28294637 0.87 ALDH1A1 (0.47) NPC1GAARAB9A
SCHEMBL28294516 0.86 KLKB1 (0.47) KLKB1KLK1PLGPRSS1NPC1
SCHEMBL28296207 0.69 NPC1 (0.44) KLKB1KLK1PLGPRSS1NPC1
SCHEMBL554803 0.68 GAA (0.60) KLKB1NPC1GAARAB9ACA12
SCHEMBL28146103 0.68 RAB9A (0.51) KLKB1KLK1NPC1POLBGAA
SCHEMBL22221787 0.67 RAB9A (0.69) NPC1POLBGAARAB9A
SCHEMBL256698 0.65
SCHEMBL28333414 0.64 LOXL2 (0.47) KLKB1KLK1NPC1POLBGAA
SCHEMBL27996204 0.64 GFER (0.70) KLKB1KLK1NPC1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106608872-B 5- pyrazol acid amide compounds and the preparation method and application thereof 湖南化工研究院有限公司 2019-04-19 CN disclosed