SCHEMBL28294579

SCHEMBL28294579

CC(=O)Nc1ccc(-c2cccc(C(=O)O)c2)cn1

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.52
ABL1 P00519 1/20 0.50
BCR P11274 1/20 0.50
PIK3CD O00329 1/20 0.49
PIK3CG P48736 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
TDO2 P48775 1/20 0.48
AXL P30530 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29128779 0.87 PTK2 (0.51) PIK3CDPIK3CGGAATDO2
SCHEMBL1553208 0.86 PIK3CA (0.65) PIK3CDPIK3CG
SCHEMBL28118455 0.84 PTK2 (0.54) PIK3CDPIK3CGGAA
SCHEMBL30338494 0.84 PTK2 (0.57) PIK3CDPIK3CGGAA
SCHEMBL23193793 0.82 BCL2 (0.48) KMOLMNAGAAAXL
SCHEMBL29627265 0.82 BCL2 (0.48) KMOLMNAGAAAXL
SCHEMBL15394357 0.80 RXRA (0.50) ABL1BCRPIK3CDPIK3CGGAA
SCHEMBL8738131 0.80 KDR (0.55) ABL1BCRPIK3CDPIK3CGGAA
SCHEMBL31055398 0.79 NAMPT (0.53) ABL1BCR
SCHEMBL5803994 0.78 ADORA2A (0.50) ABL1PIK3CDPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796439-B Hydroxyproline peptide derivative and preparation method and application thereof 西安交通大学 2020-05-19 CN claimed
CN-109796439-A A kind of hydroxyproline class peptide derivant and its preparation method and application 西安交通大学 2019-05-24 CN claimed
CN-109824582-B Alanine derivative and preparation method and application thereof 西安交通大学 2020-06-19 CN disclosed
CN-109796439-B Hydroxyproline peptide derivative and preparation method and application thereof 西安交通大学 2020-05-19 CN disclosed
CN-109824582-A A kind of alanine derivatives and its preparation method and application 西安交通大学 2019-05-31 CN disclosed
CN-109796439-A A kind of hydroxyproline class peptide derivant and its preparation method and application 西安交通大学 2019-05-24 CN disclosed