SCHEMBL28295046

SCHEMBL28295046

N#Cc1cc(N)ccc1F.Nc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 3/20 0.46
USP2 O75604 1/20 0.46
LMNA P02545 3/20 0.43
MAPT P10636 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HPGD P15428 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
GFER P55789 2/20 0.40
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
TRPV4 Q9HBA0 2/20 0.38
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KHK P50053 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30241198 0.92 KDM4E (0.52) KDM4EALDH1A1USP2LMNAMAPT
SCHEMBL145984 0.92 KDM4E (0.52) KDM4EALDH1A1USP2LMNAMAPT
Hydrochloric Acid SCHEMBL2482616 0.90 KDM4E (0.50) KDM4EALDH1A1USP2LMNAMAPT
Fluoromethane SCHEMBL28180626 0.88 KDM4E (0.53) KDM4EALDH1A1USP2LMNAMAPT
SCHEMBL21497154 0.81 CYP11B1 (0.49) ALDH1A1CYP3A4CYP11B1CYP11B2TDP1
SCHEMBL74807 0.79 TRPV4 (0.46) ALDH1A1HPGDCYP1A2CYP3A4CYP2C19
SCHEMBL1514274 0.76 CYP11B1 (0.57) ALDH1A1HPGDCYP1A2CYP3A4CYP2C19
SCHEMBL1156401 0.75 TRPV4 (0.57) KDM4EALDH1A1USP2LMNAMAPT
SCHEMBL30084909 0.75 TRPV4 (0.57) KDM4EALDH1A1USP2LMNAMAPT
SCHEMBL30084906 0.75 TRPV4 (0.57) KDM4EALDH1A1USP2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790168-A SUBSTITUTED PYRROLIZINE COMPOUNDS AND USES THEREOF 吉利德科学公司 2019-05-21 CN disclosed