SCHEMBL1156401

SCHEMBL1156401

N#Cc1ccc(N)cc1F

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.57
CYP11B2 P19099 13/20 0.54
CYP11B1 P15538 11/20 0.54
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 2/20 0.52
USP2 O75604 1/20 0.52
EGLN2 Q96KS0 1/20 0.45
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
KHK P50053 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30084906 1.00 TRPV4 (0.57) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
SCHEMBL30084909 1.00 TRPV4 (0.57) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
Fluoride SCHEMBL21646063 0.98 TRPV4 (0.55) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
Methane SCHEMBL27650148 0.98 TRPV4 (0.55) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
SCHEMBL7282150 0.84 CYP11B2 (0.66) TRPV4CYP11B2CYP11B1EGLN2
SCHEMBL30241198 0.82 KDM4E (0.52) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
SCHEMBL145984 0.82 KDM4E (0.52) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL2482616 0.80 KDM4E (0.50) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
SCHEMBL10050188 0.79 CYP19A1 (0.46) TRPV4CYP11B2CYP11B1KDM4EALDH1A1
SCHEMBL981232 0.79 CYP11B2 (0.65) TRPV4CYP11B2CYP11B1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 480 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120117998-A Preparation method of apatamide intermediate N-methyl-2-fluoro-4-aminobenzamide 成都博腾药业有限公司 2025-06-10 CN claimed
CN-114276266-B Preparation method of 4-amino-2-fluorobenzamide 兰州康鹏威耳化工有限公司 2024-10-11 CN claimed
CN-115028642-B Diaryl dihydrofuro [3,4-d ] pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2024-07-12 CN claimed
CN-116332789-A Preparation method of 4-amino-2-fluorobenzamide 上海康鹏科技股份有限公司 2023-06-27 CN claimed
CN-114276266-A Preparation method of 4-amino-2-fluorobenzamide 兰州康鹏威耳化工有限公司 2022-04-05 CN claimed
CN-108440559-B Diaryl thienopyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2020-06-16 CN claimed
CN-109678741-A The preparation method of 4- amino -3- fluobenzoic acid 金凯(辽宁)化工有限公司 2019-04-26 CN claimed
CN-108440559-A Diaryl thienopyrimidines HIV-1 reverse transcriptase inhibitor and its preparation method and application 山东大学 2018-08-24 CN claimed
JP-60163857-A None JP disclosed
US-12612383-B2 Polysubstituted pyrrolidine derivative, preparation method therefor and use thereof SHANGHAI WENNAI THERAPEUTICS CO., LTD. (CN) 2026-04-28 US disclosed
US-20260062393-A1 Compounds CTXT PTY LTD (AU) 2026-03-05 US disclosed
US-20260001886-A1 ENPP1 INHIBITORS I RE VENTURES I LLC (US) 2026-01-01 US disclosed
US-12503426-B2 Synthetic derivatives of oleoyl-lysophosphatidylinositol (oleoyl-LPI) and uses thereof LIPOVEXA SRL (IT) 2025-12-23 US disclosed
EP-4660186-A1 ACID ADDITION SALT OF 4-AMINO-2-HALOBENZONITRILE COMPOUND AND METHOD FOR PRODUCING SAME SUGAI CHEMICAL INDUSTRY CO., LTD. (JP) 2025-12-10 EP disclosed
US-4704227-A DERIVATIVES OF 1,3-DIOXANE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1987-11-03 US disclosed
EP-0154840-A2 Liquid crystal compounds MERCK PATENT GmbH (DE) 1985-09-18 EP disclosed
JP-S60163857-A SYNTHESIS OF 2-FLUORO-4-THIOBENZONITRILE HITACHI LTD 1985-08-26 JP disclosed
US-4333940-A Ring-fluorinated 4-(monosubstituted-amino) phenyl compounds in inhibiting atherosclerotic lesion development AMERICAN CYANAMID COMPANY (US) 1982-06-08 US disclosed
US-4243609-A ANTILIPEMIC AGENTS, ANTIATHEROSCLEROTIC AGENTS AMERICAN CYANAMID COMPANY (US) 1981-01-06 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503426-B2 Synthetic derivatives of oleoyl-lysophosphatidylinositol (oleoyl-LPI) and uses thereof GPR119, GLP1R, LPAR1 TRPV4 1074/4885CYP11B2 3053/4885CYP11B1 2156/4885
US-20260062393-A1 Compounds SCN2B, ABCB11, SCN1B TRPV4 1449/4885CYP11B2 629/4885CYP11B1 796/4885
US-20260001886-A1 ENPP1 INHIBITORS I ENPP1, ENPP2, ENPP3 TRPV4 4401/4885CYP11B2 1971/4885CYP11B1 1208/4885
US-12612383-B2 Polysubstituted pyrrolidine derivative, preparation method therefor and use thereof SCN8A, SCN11A, TRPV1 TRPV4 17/4885CYP11B2 1139/4885CYP11B1 1478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.