SCHEMBL28295739

SCHEMBL28295739

Cc1ccc2nccc(-c3ccc(F)cc3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.48
HTR1A P08908 2/20 0.46
ADRA1D P25100 2/20 0.46
ADRA1A P35348 2/20 0.46
ADRA1B P35368 2/20 0.46
APP P05067 1/20 0.44
GRM2 Q14416 1/20 0.44
PIK3CD O00329 2/20 0.42
PIK3CB P42338 1/20 0.42
MTOR P42345 1/20 0.42
PIK3CG P48736 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28175732 0.90 PIK3CA (0.53) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL756601 0.87 GRM2 (0.53) HTR1AADRA1DADRA1AADRA1BAPP
SCHEMBL30440111 0.85 PIK3CA (0.64) PIK3CAPIK3CDPIK3CBMTORPIK3CG
SCHEMBL28288868 0.82 MAPK14 (0.47) PIK3CAKDM4EALDH1A1AAK1GRM4
SCHEMBL28295741 0.81 TLR8 (0.51) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL28293866 0.81 PIK3CA (0.46) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL16549212 0.81 PIK3CA (0.48) PIK3CAAPPPIK3CDPIK3CBMTOR
SCHEMBL29287969 0.79 PIK3CA (0.49) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL17833787 0.77 PIK3CA (0.48) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL6660966 0.76 GRM4 (0.56) PIK3CAAAK1GRM4CCNB2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796403-B Quinoline derivatives and preparation method thereof 安徽师范大学 2021-09-28 CN disclosed
CN-109796403-A Quinoline derivatives and preparation method thereof 安徽师范大学 2019-05-24 CN disclosed