SCHEMBL28293866

SCHEMBL28293866

Cc1ccc2nccc(-c3ccc(C(C)(C)C)cc3)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.46
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.42
TSHR P16473 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KIF11 P52732 1/20 0.40
AKT1 P31749 2/20 0.38
DGAT1 O75907 2/20 0.38
ACVR1 Q04771 1/20 0.38
SLC22A12 Q96S37 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28175732 0.87 PIK3CA (0.53) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL28295739 0.81 PIK3CA (0.48) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL28925687 0.80 KDR (0.48) PIK3CAKDM4EALDH1A1MEN1KMT2A
SCHEMBL28295741 0.79 TLR8 (0.51) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL29287969 0.76 PIK3CA (0.49) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL17833787 0.75 PIK3CA (0.48) PIK3CAHTR1AADRA1DADRA1AADRA1B
SCHEMBL10154084 0.75 ACVR1 (0.49) PIK3CAMEN1KMT2AKIF11ACVR1
SCHEMBL23479555 0.74 HTR1A (0.51) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL6347874 0.74 KIF11 (0.47) ADRA1ATSHRKDM4EALDH1A1LMNA
SCHEMBL25878119 0.72 KDR (0.56) KDM4EALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796403-B Quinoline derivatives and preparation method thereof 安徽师范大学 2021-09-28 CN disclosed
CN-109796403-A Quinoline derivatives and preparation method thereof 安徽师范大学 2019-05-24 CN disclosed