SCHEMBL28295741

SCHEMBL28295741

COc1ccc(-c2ccnc3ccc(C)cc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.51
NCOA1 Q15788 1/20 0.50
NCOA3 Q9Y6Q9 1/20 0.50
DYRK1A Q13627 1/20 0.47
CYP19A1 P11511 1/20 0.46
GRM2 Q14416 1/20 0.46
SYK P43405 1/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CCNB2 O95067 1/20 0.46
CDK1 P06493 1/20 0.46
CCNB1 P14635 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
CCNB3 Q8WWL7 1/20 0.46
PIK3CA P42336 1/20 0.46
MAPT P10636 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28175732 0.87 PIK3CA (0.53) TLR8KDM4ENPSR1CCNB2CDK1
SCHEMBL16549166 0.84 CCNB2 (0.49) TLR8DYRK1AKDM4EMAPK1NPSR1
SCHEMBL16549227 0.84 MAP4K4 (0.50) TLR8DYRK1ACYP19A1SYKKDM4E
SCHEMBL28295739 0.81 PIK3CA (0.48) GRM2KDM4ENPSR1CCNB2CDK1
SCHEMBL10157305 0.80 PIK3CA (0.57) TLR8KDM4EMAPK1NPSR1PIK3CA
SCHEMBL30440258 0.80 PIK3CA (0.57) TLR8KDM4EMAPK1NPSR1PIK3CA
SCHEMBL7665284 0.80 BMP4 (0.61) TLR8SYKKDM4ENPSR1MAPT
SCHEMBL30251801 0.80 BMP4 (0.61) TLR8SYKKDM4ENPSR1MAPT
SCHEMBL28293866 0.79 PIK3CA (0.46) KDM4ENPSR1PIK3CAMAPTLMNA
SCHEMBL29287969 0.76 PIK3CA (0.49) KDM4ENPSR1PIK3CAMAPTMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796403-B Quinoline derivatives and preparation method thereof 安徽师范大学 2021-09-28 CN disclosed
CN-109796403-A Quinoline derivatives and preparation method thereof 安徽师范大学 2019-05-24 CN disclosed