SCHEMBL28296312

SCHEMBL28296312

Cc1cc(C)c(/C=C/c2ccccc2)c(/C(N)=N/c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.46
HIF1A Q16665 1/20 0.46
TTR P02766 1/20 0.41
ALOX5 P09917 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NFE2L2 Q16236 1/20 0.40
NOS1 P29475 3/20 0.40
NOS3 P29474 2/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
RAB9A P51151 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
MAPT P10636 2/20 0.37
HTR3E A5X5Y0 2/20 0.37
HTR3B O95264 2/20 0.37
HTR3A P46098 2/20 0.37
HTR3D Q70Z44 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28413170 1.00 CYP2D6 (0.46) CYP2D6HIF1ATTRALOX5PTGS1
SCHEMBL28413171 1.00 CYP2D6 (0.46) CYP2D6HIF1ATTRALOX5PTGS1
SCHEMBL698718 0.78 TTR (0.53) TTRALOX5PTGS1PTGS2NFE2L2
SCHEMBL698717 0.78 TTR (0.53) TTRALOX5PTGS1PTGS2NFE2L2
SCHEMBL28411059 0.77 CYP2D6 (0.50) CYP2D6HIF1ATTRALOX5PTGS1
SCHEMBL28296313 0.77 CYP2D6 (0.50) CYP2D6HIF1ATTRALOX5PTGS1
SCHEMBL28411058 0.77 CYP2D6 (0.50) CYP2D6HIF1ATTRALOX5PTGS1
SCHEMBL28524007 0.73 TTR (0.46) TTRALOX5PTGS1PTGS2MEN1
SCHEMBL28408255 0.72 MEN1 (0.48) CYP2D6HIF1AMEN1KMT2ANFE2L2
SCHEMBL28408254 0.72 MEN1 (0.48) CYP2D6HIF1AMEN1KMT2ANFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-B Method for preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2020-03-10 CN disclosed
CN-109796372-A A method of preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2019-05-24 CN disclosed