SCHEMBL28408255

SCHEMBL28408255

NC(=Nc1ccccc1)c1ccccc1C=Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
TRPA1 O75762 2/20 0.47
PLAU P00749 2/20 0.44
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
SLC22A2 O15244 1/20 0.44
SLC22A1 O15245 1/20 0.44
SLC22A3 O75751 1/20 0.44
NFE2L2 Q16236 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
NOS1 P29475 4/20 0.42
NOS3 P29474 2/20 0.42
CYP2D6 P10635 1/20 0.42
HIF1A Q16665 1/20 0.42
PLAT P00750 1/20 0.41
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28408256 1.00 MEN1 (0.48) MEN1KMT2ATRPA1PLAUHTR3E
SCHEMBL28408254 1.00 MEN1 (0.48) MEN1KMT2ATRPA1PLAUHTR3E
SCHEMBL28410295 0.89 NFE2L2 (0.50) MEN1KMT2ATRPA1PLAUHTR3E
SCHEMBL28410294 0.89 NFE2L2 (0.50) MEN1KMT2ATRPA1PLAUHTR3E
SCHEMBL28296333 0.89 NFE2L2 (0.50) MEN1KMT2ATRPA1PLAUHTR3E
SCHEMBL28410290 0.85 TRPA1 (0.53) TRPA1PLAUHTR3EHTR3BHTR3A
SCHEMBL28410291 0.85 TRPA1 (0.53) TRPA1PLAUHTR3EHTR3BHTR3A
SCHEMBL28296320 0.85 TRPA1 (0.53) TRPA1PLAUHTR3EHTR3BHTR3A
SCHEMBL28411059 0.82 CYP2D6 (0.50) MEN1KMT2APLAUHTR3EHTR3B
SCHEMBL28411058 0.82 CYP2D6 (0.50) MEN1KMT2APLAUHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-B Method for preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2020-03-10 CN disclosed