SCHEMBL28297921

SCHEMBL28297921

O=C1CCC(c2ccc(OC(F)F)cc2)=NN1c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
GAA P10253 2/20 0.43
HRH3 Q9Y5N1 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MT-CO2 P00403 1/20 0.39
ALDH1A1 P00352 3/20 0.39
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
BACE1 P56817 2/20 0.36
ATM Q13315 2/20 0.36
CSNK1E P49674 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297926 0.84 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DCA12
SCHEMBL19660389 0.80 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL28297934 0.80 PDCD1 (0.46) PDE4APDE4BPDE4CPDE4DCA12
SCHEMBL28299533 0.78 KDM4E (0.41) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL30187450 0.75 KDM4E (0.41) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL19642572 0.75 KDM4E (0.41) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL29395562 0.74 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DCA12
SCHEMBL29392667 0.71 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DCA12
SCHEMBL9567402 0.70 MEN1 (0.44) GAAMEN1KMT2ABACE1MAPT
SCHEMBL29394932 0.70 CA12 (0.68) PDE4APDE4BPDE4CPDE4DCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863140-A 3- oxo -2,6- diphenyl -2,3- dihydrogen dazin -4- formamide 拜耳医药股份有限公司 2019-06-07 CN disclosed