SCHEMBL28298507

SCHEMBL28298507

Fc1ccc(F)c(C2CCNC2)c1.NC=S

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
MPO P05164 1/20 0.43
KDM1A O60341 2/20 0.41
HTR3A P46098 1/20 0.41
KDM1B Q8NB78 1/20 0.41
SLC6A2 P23975 3/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A3 Q01959 3/20 0.40
HTR1A P08908 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27913713 0.91 CHRNB2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL19995723 0.91 CHRNB2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL28296873 0.83 CHRNB2 (0.44) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL28873499 0.82 HCAR2 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL1765151 0.81 SLC6A2 (0.55) CHRNB2CHRNB4CHRNA3CHRNA4HTR2A
SCHEMBL28296881 0.81 HTR3A (0.42) CHRNB2CHRNB4CHRNA3CHRNA4HTR2C
SCHEMBL28298501 0.80 HTR3A (0.56) HTR2CMPOHTR3A
Hydrochloric Acid SCHEMBL6075890 0.79 SLC6A2 (0.54) CHRNB2CHRNB4CHRNA3CHRNA4HTR2C
SCHEMBL28298496 0.79 HTR3A (0.51) HTR2CKDM1AHTR3ASLC6A2SLC6A4
SCHEMBL1822160 0.78 CHRNB2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed