SCHEMBL28296881

SCHEMBL28296881

Fc1ccc(C2CCNC2)c(F)c1F.NC=S

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.42
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
HTR1A P08908 1/20 0.38
CYP2D6 P10635 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19995543 0.91 HTR3A (0.46) HTR3ACHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL7380797 0.81 HTR2A (0.46) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL28298507 0.81 CHRNB2 (0.44) HTR3ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL10419750 0.80 SLC6A2 (0.48) SLC6A2SLC6A4HTR1ASLC6A3HTR2C
SCHEMBL1824314 0.79 CHRNB2 (0.49) CHRNB2CHRNA7CHRNA4SLC6A2SLC6A4
SCHEMBL28296873 0.78 CHRNB2 (0.44) HTR3ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL28873499 0.78 HCAR2 (0.38) HTR3ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL28298496 0.77 HTR3A (0.51) HTR3ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL20438982 0.75 KDM1A (0.40) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL28296852 0.75 HTR3A (0.38) HTR3ACHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed