SCHEMBL28298884

SCHEMBL28298884

COc1cccc(C(=O)Nc2c(C(N)=O)cnc3c(C)cccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
NPSR1 Q6W5P4 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HPGD P15428 1/20 0.53
MAPK10 P53779 1/20 0.53
HSD17B10 Q99714 1/20 0.53
AURKA O14965 1/20 0.52
RPS6KB1 P23443 1/20 0.52
AURKB Q96GD4 1/20 0.52
PDE4B Q07343 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
GRM5 P41594 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2635973 0.83 PDE4B (0.73) PDE4BTP53
SCHEMBL28298882 0.82 TSHR (0.50) TSHRNPSR1MEN1KMT2AHPGD
SCHEMBL13754028 0.73 PDE4B (0.73) PDE4B
SCHEMBL27568903 0.73 CSF1R (0.71)
SCHEMBL21870539 0.72 TSHR (0.66) TSHRNPSR1MEN1KMT2AHPGD
SCHEMBL18912123 0.71 PDE4B (0.62) PDE4B
SCHEMBL1311332 0.71 PDE4B (0.71) PDE4BTP53
SCHEMBL18343125 0.71 ALDH1A1 (0.61) TSHRNPSR1MEN1KMT2ASMN1; SMN2
SCHEMBL259608 0.71 ALDH1A1 (0.61) TSHRNPSR1MEN1KMT2ASMN1; SMN2
SCHEMBL882567 0.71 MEN1 (0.76) TSHRNPSR1MEN1KMT2AMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109789150-A It is certain to be used to treat bronchiectasic (2S)-N- [(1S) -1- cyano -2- phenethyl] -1,4- oxazepine cycloheptane -2- formamide 英斯梅德股份有限公司 2019-05-21 CN disclosed