SCHEMBL28298882

SCHEMBL28298882

COc1cccc(C(=O)Nc2c(NC=O)cnc3c(C)cccc23)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
NPSR1 Q6W5P4 2/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
GRM5 P41594 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TP53 P04637 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28298884 0.82 TSHR (0.53) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL21870539 0.71 TSHR (0.66) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL29808279 0.71 MEN1 (0.83) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL12077495 0.71 MEN1 (0.83) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL11246385 0.68 MEN1 (1.00) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL13319566 0.67 MEN1 (0.65) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL6537714 0.67 KMT2A (0.61) SMN1; SMN2MEN1KMT2AALDH1A1LMNA
SCHEMBL21829023 0.67 KMT2A (0.78) SMN1; SMN2MEN1KMT2AALDH1A1LMNA
SCHEMBL277650 0.66 ALDH1A1 (0.61) TSHRNPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL277775 0.66 ALDH1A1 (0.61) TSHRNPSR1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109789150-A It is certain to be used to treat bronchiectasic (2S)-N- [(1S) -1- cyano -2- phenethyl] -1,4- oxazepine cycloheptane -2- formamide 英斯梅德股份有限公司 2019-05-21 CN disclosed