SCHEMBL28299864

SCHEMBL28299864

O=C(On1cccc1)c1ncccc1OC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.41
HCRTR1 O43613 3/20 0.40
DHODH Q02127 1/20 0.37
HCRTR2 O43614 1/20 0.36
SSTR1 P30872 3/20 0.36
SSTR4 P31391 3/20 0.36
HSD17B13 Q7Z5P4 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
GAA P10253 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
HCAR1 Q9BXC0 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34
NFE2L2 Q16236 1/20 0.34
ATR Q13535 1/20 0.34
CYP2C9 P11712 1/20 0.34
EPHX2 P34913 1/20 0.34
CYP2J2 P51589 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31471005 0.80 L3MBTL1 (0.53) TLR7HCRTR1DHODHHCRTR2SSTR1
SCHEMBL30368262 0.77 KDM4E (0.50) TLR7HCRTR1DHODHHCRTR2HSD17B13
SCHEMBL2301103 0.77 KDM4E (0.50) TLR7HCRTR1DHODHHCRTR2HSD17B13
SCHEMBL15142683 0.76 SMN1; SMN2 (0.45) TLR7HCRTR1HCRTR2HSD17B13ADORA2A
SCHEMBL31307011 0.76 BRD4 (0.53) TLR7HCRTR1P2RY1
SCHEMBL28152819 0.75 CASP3 (0.38) GAA
SCHEMBL16571480 0.70 HCRTR1 (0.40) TLR7HCRTR1DHODHHCRTR2HSD17B13
SCHEMBL28102316 0.69 HCRTR1 (0.41) HCRTR1HCRTR2GAA
SCHEMBL13419577 0.68 SLC40A1 (0.40) DHODHRXRARXRBRXRGSLC40A1
SCHEMBL17506347 0.68 TLR7 (0.40) TLR7HCRTR1HSD17B13ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109956929-A Hete rocyclic derivatives, preparation method, pharmaceutical composition and application 上海迪诺医药科技有限公司 2019-07-02 CN disclosed