SCHEMBL28301495

SCHEMBL28301495

COc1ccc(NC(=O)C#Cc2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 1.00
NPC1 O15118 7/20 1.00
KMT2A Q03164 3/20 1.00
MEN1 O00255 2/20 1.00
POLB P06746 1/20 1.00
NLRP3 Q96P20 1/20 1.00
ALDH1A1 P00352 4/20 0.57
MAPT P10636 4/20 0.57
CYP1A2 P05177 3/20 0.57
CYP2C19 P33261 3/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2C9 P11712 2/20 0.57
TSHR P16473 1/20 0.57
GFER P55789 1/20 0.54
VCP P55072 1/20 0.53
SMN1; SMN2 Q16637 5/20 0.53
HTT P42858 2/20 0.53
GAA P10253 1/20 0.53
CYP2D6 P10635 1/20 0.52
METAP2 P50579 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30056033 0.94 RAB9A (0.89) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL1250 0.84 NPC1 (0.71) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL9263110 0.83 NPC1 (0.70) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL9820160 0.82 RAB9A (0.69) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL3857350 0.80 KMT2A (0.66) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL28302925 0.80 MEN1 (0.66) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL6241316 0.79 NPC1 (0.65) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL22462232 0.79 RAB9A (0.65) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL13847795 0.78 NPC1 (0.64) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL14336956 0.78 RAB9A (0.63) RAB9ANPC1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110066254-A A kind of isothiazole -3- ketone compound and preparation method thereof 温州大学 2019-07-30 CN disclosed
CN-110054597-A A kind of thiazolidin-4-one derivatives and preparation method thereof synthesized under the conditions of non-metal catalyst 温州大学 2019-07-26 CN disclosed
CN-109796423-A The method of 1,3- thiazine -4- ketone is synthesized under no metal catalyzed conditions 温州大学 2019-05-24 CN disclosed