SCHEMBL9820160

SCHEMBL9820160

COc1ccc(NC(=S)C#Cc2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.69
NPC1 O15118 4/20 0.69
KMT2A Q03164 3/20 0.69
MEN1 O00255 2/20 0.69
POLB P06746 1/20 0.69
NLRP3 Q96P20 1/20 0.69
CYP1A2 P05177 3/20 0.59
CYP2C19 P33261 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.56
MAPT P10636 6/20 0.55
ALDH1A1 P00352 4/20 0.55
HTT P42858 1/20 0.55
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 2/20 0.53
TSHR P16473 2/20 0.51
MAOB P27338 3/20 0.50
MAOA P21397 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
HPGD P15428 1/20 0.49
GAA P10253 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28301495 0.82 RAB9A (1.00) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL30056033 0.76 RAB9A (0.89) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL1259295 0.75 CYP1A2 (1.00) RAB9ANPC1KMT2AMEN1CYP1A2
Hydrogen Sulfide SCHEMBL28246712 0.74 CYP1A2 (0.96) RAB9ANPC1KMT2AMEN1CYP1A2
SCHEMBL7306947 0.73 CYP1A2 (0.69) RAB9ANPC1KMT2AMEN1CYP1A2
SCHEMBL1180922 0.72 NPC1 (1.00) RAB9ANPC1KMT2AMEN1CYP1A2
SCHEMBL6241316 0.72 NPC1 (0.65) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL28953063 0.72 NPC1 (0.56) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL5552160 0.72 APP (0.65) RAB9ANPC1KMT2AMEN1POLB
Fluoride SCHEMBL28392203 0.71 CYP1A2 (0.67) RAB9ANPC1KMT2AMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248523-B1 PYRAZOLES FISONS plc (GB) 1991-10-16 EP disclosed
US-4803216-A Pyrazole-3-amines as anti-inflammatory agents FISONS PLC (GB) 1989-02-07 US disclosed
EP-0248523-A1 Pyrazoles FISONS plc (GB) 1987-12-09 EP disclosed