SCHEMBL2830187

SCHEMBL2830187

CC=CNc1cc[nH]c(=O)n1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830185 1.00 ADORA2A (0.33) ADORA2AADORA1DYRK1A
SCHEMBL5841377 0.80 ALDH1A1 (0.32) ADORA2AADORA1DYRK1A
SCHEMBL29752139 0.79 NPC1 (0.36) DYRK1A
SCHEMBL4306636 0.78 DYRK1A (0.31) ADORA2AADORA1DYRK1A
SCHEMBL27952254 0.75 NCF1 (0.39) ADORA2AADORA1DYRK1A
SCHEMBL10865972 0.75 ADORA2A (0.30) ADORA2AADORA1
Hydrochloric Acid SCHEMBL6853662 0.74 NCF1 (0.38) ADORA2AADORA1DYRK1A
SCHEMBL30917959 0.74 NCF1 (0.38) ADORA2AADORA1DYRK1A
SCHEMBL8080125 0.72 ADORA2A (0.35) ADORA2AADORA1DYRK1A
SCHEMBL8944768 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874790-B1 NEW S-ADENOSYL-L-METHIONINE ANALOGS WITH EXTENDED ACTIVATED GROUPS FOR TRANSFER BY METHYLTRANSFERASES RWTH AACHEN (DE) 2010-08-18 EP disclosed
EP-1874790-A2 NEW S-ADENOSYL-L-METHIONINE ANALOGS WITH EXTENDED ACTIVATED GROUPS FOR TRANSFER BY METHYLTRANSFERASES RWTH Aachen (DE) 2008-01-09 EP disclosed
WO-2006108678-A2 NEW S-ADENOSYL-L-METHIONINE ANALOGS WITH EXTENDED ACTIVATED GROUPS FOR TRANSFER BY METHYLTRANSFERASES RWTH AACHEN (DE) 2006-10-19 WO disclosed
EP-1712557-A1 New s-adenosyl-L-methionine analogues with extended activated groups for transfer by methyltransferases RWTH Aachen (DE) 2006-10-18 EP disclosed