SCHEMBL2830652

SCHEMBL2830652

CN(C)C1(c2ccccc2F)CCC(=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC4 P56524 2/20 0.38
OPRM1 P35372 4/20 0.37
OPRL1 P41146 4/20 0.37
OPRK1 P41145 2/20 0.37
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.34
RECQL P46063 1/20 0.34
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
HCAR2 Q8TDS4 1/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11096498 0.81 MEN1 (0.40) CYP2C9MEN1KMT2AHDAC4OPRM1
Iodide SCHEMBL11093787 0.79 MEN1 (0.39) CYP2C9MEN1KMT2AHDAC4OPRM1
SCHEMBL11094080 0.79 GRIN1 (0.45) CYP2C9MEN1KMT2AHDAC4OPRM1
SCHEMBL9729622 0.78 MEN1 (0.53) CYP2C9MEN1KMT2AHDAC4OPRM1
SCHEMBL11096692 0.78 CYP2D6 (0.42) CYP2C9MEN1KMT2AHDAC4OPRM1
Ethylene SCHEMBL11093850 0.78 MEN1 (0.38) CYP2C9MEN1KMT2AHDAC4OPRM1
SCHEMBL11096483 0.77 SLC6A3 (0.47) CYP2C9MEN1KMT2AOPRM1OPRL1
SCHEMBL6952827 0.75 OPRM1 (0.50) CYP2C9MEN1KMT2AHDAC4OPRM1
SCHEMBL17982791 0.75 MEN1 (0.41) CYP2C9MEN1KMT2AHDAC4PSEN1
SCHEMBL11559606 0.75 HDAC4 (0.41) CYP2C9MEN1KMT2AHDAC4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233487-A1 Spirocyclic cyclohexane derivatives Grünenthal GmbH (DE) 2010-09-29 EP disclosed