SCHEMBL2830666

SCHEMBL2830666

C=C(OCCCC)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
LMNA P02545 4/20 0.42
TSHR P16473 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
MAPK1 P28482 2/20 0.42
ESR1 P03372 2/20 0.42
CYP2D6 P10635 1/20 0.42
NR1H2 P55055 1/20 0.42
RNASEL Q05823 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PDE4D Q08499 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21836017 0.81 HDAC3 (0.48) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12251325 0.80 ESR1 (0.68) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7695874 0.79 TSHR (0.45) LMNATSHRSMN1; SMN2CYP1A2CYP2C19
SCHEMBL2539792 0.79 TSHR (0.50) LMNATSHRSMN1; SMN2CYP1A2CYP2C19
SCHEMBL5710014 0.74 ALDH1A1 (0.68) HDAC3HDAC1HDAC2LMNATSHR
SCHEMBL1322179 0.74 ALDH1A1 (0.68) HDAC3HDAC1HDAC2LMNATSHR
SCHEMBL11330183 0.74 ALDH1A1 (0.68) HDAC3HDAC1HDAC2LMNATSHR
SCHEMBL29032300 0.74 ALDH1A1 (0.68) HDAC3HDAC1HDAC2LMNATSHR
SCHEMBL25013199 0.73 ALDH1A1 (0.67) LMNATSHRCYP1A2CYP2C19CYP2D6
SCHEMBL8029452 0.73 PKM (0.49) HDAC3HDAC1HDAC2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8435387-B2 Small-scale method and apparatus for separating mixtures MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2013-05-07 US disclosed
US-20100122899-A1 SMALL-SCALE METHOD AND APPARATUS FOR SEPARATING MIXTURES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-05-20 US disclosed
WO-2010056331-A2 SMALL-SCALE METHOD AND APPRATUS FOR SEPARATING MIXTURES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-05-20 WO disclosed