SCHEMBL28308550

SCHEMBL28308550

CC(C)(C)c1c(C#N)c(Cl)nc2c1CNCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.44
MAPK1 P28482 1/20 0.44
KDM4E B2RXH2 2/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
HTT P42858 4/20 0.35
GLA P06280 1/20 0.35
ALDH1A1 P00352 4/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PDE5A O76074 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
MAPT P10636 1/20 0.31
PNMT P11086 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24891788 0.71 HTT (0.46) NSD2MAPK1KDM4EHTR2AHTR2C
SCHEMBL1119947 0.66 PNMT (0.39) HTR2AHTR2CHTR2BMAPTPNMT
SCHEMBL24892162 0.65 HTT (0.42) NSD2MAPK1KDM4EHTR2BHTT
SCHEMBL30501086 0.65 MAPK1 (0.66) NSD2MAPK1KDM4EHTTGLA
SCHEMBL23783191 0.65 MAPK1 (0.66) NSD2MAPK1KDM4EHTTGLA
SCHEMBL17985355 0.65 SMN1; SMN2 (0.62) KDM4EHTR2AHTR2CHTR2BALDH1A1
SCHEMBL24891984 0.65 KDM4E (0.38) NSD2MAPK1KDM4EHTR2AHTR2C
SCHEMBL12706725 0.64 HTR2A (0.49) HTR2AHTR2CHTR2BMAPTPNMT
SCHEMBL2572051 0.63 PNMT (0.42) HTR2AHTR2CHTR2BMAPTPNMT
SCHEMBL416988 0.62 PNMT (0.41) HTR2AHTR2CHTR2BMAPTPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207532-B Nitroimidazole derivatives against tuberculosis 南京明德新药研发股份有限公司 2019-07-30 CN disclosed