SCHEMBL28308809

SCHEMBL28308809

N#Cc1ccccc1-c1ccc(-n2cccn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
NOTUM Q6P988 1/20 0.47
NR3C1 P04150 1/20 0.47
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 2/20 0.44
KDM4E B2RXH2 1/20 0.44
EDNRB P24530 1/20 0.41
EDNRA P25101 1/20 0.41
CHRM1 P11229 1/20 0.41
TBK1 Q9UHD2 1/20 0.41
PTPN5 P54829 1/20 0.40
GRM5 P41594 2/20 0.40
TRPA1 O75762 1/20 0.40
PDK2 Q15119 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA10 Q9GZZ6 1/20 0.39
CHRNA9 Q9UGM1 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19794397 0.79 NOTUM (0.55) NOTUMALDH1A1MAPK1KDM4EEDNRB
SCHEMBL16388509 0.78 NR3C1 (0.42) ESR2NR3C1ALDH1A1MAPK1KDM4E
SCHEMBL16371342 0.77 ADORA2A (0.43) NOTUMALDH1A1MAPK1KDM4EEDNRB
SCHEMBL21289803 0.76 NOTUM (0.51) NOTUMALDH1A1MAPK1KDM4EEDNRB
SCHEMBL44890 0.75 NOTUM (0.58) NOTUMALDH1A1MAPK1KDM4EGRM5
SCHEMBL22030032 0.75 NOTUM (0.50) NOTUMALDH1A1MAPK1KDM4EEDNRB
SCHEMBL514359 0.75 NOTUM (0.62) NOTUMALDH1A1MAPK1KDM4ECHRM1
SCHEMBL31410710 0.74 ESR2 (0.76) ESR2ALDH1A1MAPK1KDM4EPTPN5
SCHEMBL4341894 0.74 NOTUM (0.78) NOTUMALDH1A1MAPK1KDM4ECHRM1
SCHEMBL29563253 0.74 NPC1 (0.51) NOTUMALDH1A1MAPK1KDM4EGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105517999-B IDO inhibitors 百时美施贵宝公司 2019-06-28 CN disclosed