SCHEMBL28309154

SCHEMBL28309154

COC(=O)C(OC(F)(F)F)C(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
TSHR P16473 2/20 0.43
SRC P12931 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
ROCK2 O75116 1/20 0.40
GAA P10253 1/20 0.39
CES1 P23141 2/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
CES2 O00748 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27721289 0.77 CES1 (0.50) KMT2ATSHRSRCPTGS1PTGS2
SCHEMBL31423404 0.76 MAPT (0.44) KMT2ATSHRCES1ALDH1A1CYP3A4
SCHEMBL16453798 0.75 KMT2A (0.53) KMT2ATSHRPTGS1PTGS2GAA
SCHEMBL7735376 0.75 KMT2A (0.53) KMT2ATSHRPTGS1PTGS2GAA
SCHEMBL6618828 0.74 KMT2A (0.51) KMT2ATSHRSRCPTGS1PTGS2
SCHEMBL1932808 0.73 CES1 (0.46) KMT2ATSHRSRCCES1ALDH1A1
SCHEMBL7724578 0.73 TDP1 (0.44) KMT2ATSHRCES1ALDH1A1CYP3A4
SCHEMBL2097359 0.73 KMT2A (0.55) KMT2ATSHRSRCPTGS1PTGS2
SCHEMBL8845741 0.73 KMT2A (0.55) KMT2ATSHRSRCPTGS1PTGS2
SCHEMBL27293692 0.73 KMT2A (0.49) KMT2ATSHRALDH1A1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110066236-B 1H-pyrrole derivative, preparation method thereof, pharmaceutical composition and application thereof 上海迪诺医药科技有限公司 2023-03-24 CN disclosed
CN-110066236-A 1H- azole derivatives, preparation method, pharmaceutical composition and application 上海迪诺医药科技有限公司 2019-07-30 CN disclosed