SCHEMBL28310779

SCHEMBL28310779

C=CC(=O)Nc1cccc(OCCOC)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.58
BTK Q06187 8/20 0.58
ITK Q08881 5/20 0.58
JAK2 O60674 1/20 0.58
LYN P07948 1/20 0.58
TEC P42680 1/20 0.58
TXK P42681 1/20 0.58
BMX P51813 1/20 0.58
JAK3 P52333 1/20 0.58
CD69 Q07108 1/20 0.58
MAP2K7 O14733 1/20 0.53
THRB P10828 1/20 0.52
TGM2 P21980 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14707651 0.85 EGFR (0.59) EGFRBTKITKMAP2K7THRB
SCHEMBL5037362 0.85 MAP2K7 (0.59) EGFRITKMAP2K7THRBTGM2
SCHEMBL28310060 0.83 TGM2 (0.67) EGFRBTKITKJAK2LYN
SCHEMBL1383792 0.83 TGM2 (0.66) EGFRITKTGM2
SCHEMBL31069810 0.83 TGM2 (0.66) EGFRITKTGM2
SCHEMBL12518303 0.82 EGFR (0.88) EGFRBTKITKJAK2LYN
SCHEMBL30935137 0.80 TGM2 (0.47) EGFRBTKITKJAK2LYN
SCHEMBL28463718 0.80 EGFR (0.63) EGFRBTKITKJAK2LYN
SCHEMBL30935289 0.78 BTK (0.43) EGFRBTKITKJAK2LYN
SCHEMBL184081 0.78 TP53 (0.56) EGFRBTKITKMAP2K7TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041331-B Styrylxanthine derivative and use thereof 广东东阳光药业有限公司 2020-08-07 CN disclosed
CN-110041331-A Styryl xanthine derivative and application thereof 广东东阳光药业有限公司 2019-07-23 CN disclosed