SCHEMBL28313759

SCHEMBL28313759

COc1c(OC)c2ccccc2c2ccccc12.N#CC#N

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.64
ALDH1A1 P00352 5/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
MAPK1 P28482 1/20 0.64
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 1/20 0.48
IDO1 P14902 1/20 0.48
POLB P06746 1/20 0.45
IMPDH2 P12268 1/20 0.44
IMPDH1 P20839 1/20 0.44
SLC2A1 P11166 1/20 0.40
CYP2C19 P33261 1/20 0.39
MCL1 Q07820 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL757747 0.87 KDM4E (0.82) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL8859782 0.82 ALDH1A1 (0.82) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL4958710 0.79 KDM4E (0.61) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL31171419 0.79 KDM4E (0.61) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL52405 0.79 ALDH1A1 (1.00) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL29366129 0.79 ALDH1A1 (1.00) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
Iodide SCHEMBL5967814 0.76 ALDH1A1 (0.94) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL1128021 0.76 KDM4E (0.64) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL22788818 0.73 KDM4E (0.67) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL18950744 0.73 KDM4E (0.75) KDM4EALDH1A1SMN1; SMN2MAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110156988-A A kind of phenanthro- imidazole radicals aerotex and its preparation method and application 湘潭大学 2019-08-23 CN claimed
CN-110156988-A A kind of phenanthro- imidazole radicals aerotex and its preparation method and application 湘潭大学 2019-08-23 CN disclosed