SCHEMBL28313996

SCHEMBL28313996

O=CNc1nc[nH]c(=O)c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 1/20 0.39
MCL1 Q07820 1/20 0.39
ALDH1A1 P00352 1/20 0.36
PARP1 P09874 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
ADORA2A P29274 1/20 0.34
SLC6A4 P31645 1/20 0.34
ADRA1A P35348 1/20 0.34
XDH P47989 1/20 0.34
RAB9A P51151 1/20 0.34
BLM P54132 1/20 0.34
PNP P00491 5/20 0.32
PDPK1 O15530 2/20 0.32
ACHE P22303 1/20 0.32
GDA Q9Y2T3 1/20 0.32
CA12 O43570 1/20 0.32
ALOX15 P16050 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16079874 0.79
SCHEMBL29289347 0.74 PARP1 (0.39) BCL2MCL1ALDH1A1PARP1SMN1; SMN2
SCHEMBL8426937 0.72 KDM4E (0.30) ALDH1A1SMN1; SMN2HPGD
SCHEMBL18838194 0.71 PARP1 (0.42) BCL2MCL1ALDH1A1PARP1SMN1; SMN2
SCHEMBL13348706 0.71
SCHEMBL13348604 0.68
SCHEMBL28267847 0.67 PARP1 (0.32) PARP1
SCHEMBL24161202 0.66
SCHEMBL12138872 0.66
SCHEMBL2787049 0.65 ALDH1A1 (0.32) ALDH1A1SMN1; SMN2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110214142-A It can be used as four ring heterocyclic compounds of hiv integrase inhibitor 默沙东公司 2019-09-06 CN disclosed
CN-110062627-A Tricyclic heterocyclic compounds useful as HIV integrase inhibitors 默沙东公司 2019-07-26 CN disclosed