SCHEMBL28314005

SCHEMBL28314005

Cc1ccc(C(O)=S)c(C)c1C#N

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 4/20 0.33
ALOX15 P16050 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 5/20 0.32
HPGD P15428 2/20 0.32
MAPT P10636 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.32
NOTUM Q6P988 2/20 0.31
GAA P10253 3/20 0.31
GRM6 O15303 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
UPP1 Q16831 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3107355 0.81 NOTUM (0.40) CYP1A2KDM4EALOX15HSD17B10ALDH1A1
SCHEMBL28992453 0.76 KDM4E (0.36) CYP1A2CYP2C19KDM4EALOX15HSD17B10
SCHEMBL28452345 0.74 TRPA1 (0.32) CYP1A2ALDH1A1MAPT
SCHEMBL19914848 0.74 CYP1A2 (0.42) CYP1A2CYP2C19KDM4EALOX15HSD17B10
SCHEMBL28315220 0.73 ALDH1A1 (0.48) CYP1A2CYP2C19KDM4EHSD17B10ALDH1A1
SCHEMBL31050110 0.71 CYP1A2 (0.46) CYP1A2CYP2C19KDM4EALOX15HSD17B10
SCHEMBL7975208 0.71 CYP1A2 (0.46) CYP1A2CYP2C19KDM4EALOX15HSD17B10
SCHEMBL11773357 0.69
SCHEMBL27950382 0.69 POLB (0.48) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL8852021 0.69 TSHR (0.44) CYP1A2CYP2C19KDM4EALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110183392-B Preparation method of 3-substituted phenyl-4, 5-dihydroisoxazole derivative, application and intermediate thereof 河北医科大学 2023-03-28 CN disclosed
CN-110183392-A A kind of preparation method and its usage and intermediate of 3- substituted-phenyl -4,5- dihydro-isoxazole derivative 河北医科大学 2019-08-30 CN disclosed