SCHEMBL28316282

SCHEMBL28316282

Cc1ccc(-n2c(C=O)nnc2C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2C9 P11712 4/20 0.36
CYP2C19 P33261 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALDH1A1 P00352 4/20 0.35
ALPG P10696 1/20 0.35
GAA P10253 1/20 0.34
HPGD P15428 3/20 0.33
HSP90AA1 P07900 2/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8287013 0.76 KDM4E (0.41) KDM4EALOX15TSHRL3MBTL1CYP2C9
SCHEMBL11996161 0.76 KDM4E (0.41) KDM4EALOX15TSHRL3MBTL1CYP2C9
SCHEMBL28726393 0.75 CYP1A2 (0.46) CYP1A2ALDH1A1GAAHTTPTGS2
SCHEMBL28726409 0.67 L3MBTL1 (0.52) KDM4EL3MBTL1CYP2C9CYP2C19CYP1A2
SCHEMBL11594068 0.65 AVPR1A (0.51) KDM4EALOX15TSHRMEN1KMT2A
SCHEMBL11277462 0.65 AVPR1A (0.51) KDM4ETSHRMEN1KMT2AALDH1A1
SCHEMBL27567953 0.65 KDM4E (0.40) KDM4EALOX15TSHRL3MBTL1CYP2C9
SCHEMBL5445031 0.64 TDP1 (0.63) KDM4EMEN1KMT2ACYP1A2CYP3A4
SCHEMBL5551503 0.64 ALDH1A1 (0.70) KDM4EL3MBTL1CYP2C9CYP2C19MEN1
SCHEMBL23877034 0.63 PTGER4 (0.41) KDM4EALOX15TSHRL3MBTL1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110194749-A 3- trifluoro (difluoro) methyl-1, the synthetic method of 2,4- triazole -5- ketone compounds 福州大学 2019-09-03 CN disclosed