SCHEMBL28320690

SCHEMBL28320690

C[C@@H]1CN(OC(=O)C(C)(C)C)CCN1CC1CC1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.31
CNR2 P34972 1/20 0.30
NR1H2 P55055 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28776242 0.80 DRD3 (0.30)
SCHEMBL28721922 0.74 NR1H2 (0.48) NR1H2
SCHEMBL28721924 0.74 NR1H2 (0.48) NR1H2
SCHEMBL28938073 0.74 NR1H2 (0.48) NR1H2
SCHEMBL28458593 0.72 TSHR (0.33)
SCHEMBL28876754 0.71 NR1H2 (0.30) NR1H2
SCHEMBL18701954 0.71 SPR (0.39) CNR2
SCHEMBL4698579 0.70 CHRM2 (0.36)
SCHEMBL4399555 0.70 CHRM2 (0.36)
SCHEMBL28721334 0.69 CHRM1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-A Quinazolinones PARP-1 inhibitor and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2019-08-02 CN disclosed