SCHEMBL28330968

SCHEMBL28330968

COc1ccc(CNc2ccc(C(=O)OOC(C)(C)C)cc2)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
HIF1A Q16665 3/20 0.47
APLNR P35414 1/20 0.47
KDM4C Q9H3R0 1/20 0.45
DHFR P00374 1/20 0.44
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C19 P33261 3/20 0.44
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
USP2 O75604 1/20 0.44
NAMPT P43490 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21639588 0.88 CA1 (0.58) CA1CA2HIF1AAPLNRKDM4C
SCHEMBL21639656 0.82 CA1 (0.72) CA1CA2HIF1AAPLNRKDM4C
SCHEMBL28332205 0.80 KDM4C (0.51) HIF1AAPLNRKDM4CCYP1A2CYP3A4
SCHEMBL27948920 0.78 APLNR (0.69) HIF1AAPLNRDHFRALDH1A1HSD17B10
SCHEMBL20132420 0.77 CA1 (0.76) CA1CA2HIF1AALDH1A1USP2
SCHEMBL468287 0.75 HSD17B10 (0.65) CA1CA2CYP1A2CYP2C19ALDH1A1
SCHEMBL15400259 0.73 APLNR (0.61) HIF1AAPLNRDHFRCYP1A2CYP3A4
SCHEMBL11983159 0.73 APLNR (0.65) HIF1AAPLNRDHFRCYP1A2CYP3A4
SCHEMBL28124357 0.73 CA1 (0.69) CA1CA2HIF1ACYP1A2ALDH1A1
SCHEMBL28123909 0.72 CA1 (0.59) CA1CA2HIF1AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110446699-A 2(1H) -quinolinone derivatives TAISHO PHARMACEUTICAL CO LTD 2019-11-12 CN disclosed