SCHEMBL28333141

SCHEMBL28333141

CC(C)(C)OC(=O)C1=CC=CNC(C(=O)O)=N1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28333042 0.79
SCHEMBL4334920 0.71 ALDH1A1 (0.30) ALDH1A1LMNA
SCHEMBL27517433 0.69 CA12 (0.33) ALDH1A1LMNACA12CA1CA2
SCHEMBL28105511 0.68
SCHEMBL2343974 0.67 CYP2C9 (0.34) ALDH1A1LMNACA12CA1CA2
SCHEMBL6193368 0.65 CA12 (0.34) ALDH1A1CA12CA1CA2CA9
SCHEMBL10815505 0.64 CA12 (0.35) ALDH1A1LMNACA12CA1CA2
SCHEMBL28273227 0.64 GABRA1 (0.33) CA12CA1CA2CA9CA14
SCHEMBL1615450 0.62 ELANE (0.33) ALDH1A1LMNACA12CA1CA2
SCHEMBL4334916 0.62 CA12 (0.32) ALDH1A1LMNACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110551129-B Preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester 常州合全药业有限公司 2021-11-09 CN claimed
CN-110551129-A preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester CHANGZHOU STA PHARMACEUTICAL CO LTD 2019-12-10 CN claimed
CN-110551129-B Preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester 常州合全药业有限公司 2021-11-09 CN disclosed
CN-110551129-B Preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester 常州合全药业有限公司 2021-11-09 CN disclosed
CN-110551129-B Preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester 常州合全药业有限公司 2021-11-09 CN disclosed
CN-110551129-A preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester CHANGZHOU STA PHARMACEUTICAL CO LTD 2019-12-10 CN disclosed
CN-110551129-A preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester CHANGZHOU STA PHARMACEUTICAL CO LTD 2019-12-10 CN disclosed
CN-110551129-A preparation method of 4, 5-dihydro-1H, 3H-pyrrolo [1,2-A ] [1,4] diazepine-2, 4-dicarboxylic acid-2-tert-butyl ester CHANGZHOU STA PHARMACEUTICAL CO LTD 2019-12-10 CN disclosed