SCHEMBL28338583

SCHEMBL28338583

COc1ccc(-c2nnn(Cc3ccccc3)c2-c2cccs2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.58
KMT2A Q03164 1/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 1/20 0.45
TOP2A P11388 1/20 0.45
PDE10A Q9Y233 1/20 0.45
IDO1 P14902 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NR1H4 Q96RI1 1/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MGAM O43451 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28340574 0.88 CDC7 (0.64) CDC7KMT2APOLBIDO1CYP1A2
SCHEMBL4288995 0.75 CDC7 (0.58) CDC7KMT2AIDO1
SCHEMBL4286371 0.74 CDC7 (1.00) CDC7
SCHEMBL24570328 0.73 RAB9A (0.53) CDC7NPC1RAB9AL3MBTL1POLB
SCHEMBL24570374 0.71 NPC1 (0.51) CDC7KMT2ANPC1RAB9AL3MBTL1
SCHEMBL25269369 0.71 MAPK14 (0.61) CDC7KMT2APOLBTOP2AIDO1
SCHEMBL2898117 0.71 IDO1 (0.65) CDC7POLBIDO1ALDH1A1TSHR
SCHEMBL3667857 0.70 CDC7 (0.83) CDC7
SCHEMBL21313236 0.69 ALDH1A1 (0.51) NPC1RAB9AL3MBTL1PDE10ACYP2D6
SCHEMBL6361740 0.69 P2RX7 (0.65) KMT2ANPC1RAB9AL3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110590685-A Preparation method and application of novel 5-thiocyanate substituted 1,4, 5-trisubstituted 1,2, 3-triazole 大连理工大学 2019-12-20 CN disclosed