SCHEMBL28340992

SCHEMBL28340992

Clc1ccc2c(c1)C(c1ccccc1)=NCC2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 5/20 0.58
OPRK1 P41145 5/20 0.56
PDE4D Q08499 3/20 0.56
NR1I2 O75469 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
HTR2C P28335 1/20 0.56
ADRA1A P35348 1/20 0.56
PTGS2 P35354 1/20 0.56
CHRNA4 P43681 1/20 0.56
SLC6A3 Q01959 1/20 0.56
MAPK9 P45984 1/20 0.51
MAPK14 Q16539 1/20 0.51
CNR1 P21554 2/20 0.49
NTSR1 P30989 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CHRM1 P11229 1/20 0.49
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
GABRA1 P14867 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27601351 0.93 MAPK10 (0.52) MAPK10OPRK1PDE4DNR1I2ADORA3
SCHEMBL5347707 0.91 OPRK1 (0.53) MAPK10OPRK1PDE4DNR1I2ADORA3
Hydrochloric Acid SCHEMBL11001196 0.89 OPRK1 (0.52) MAPK10OPRK1PDE4DNR1I2ADORA3
SCHEMBL8215360 0.87 MAPK10 (0.62) MAPK10OPRK1PDE4DNR1I2ADORA3
SCHEMBL6718309 0.84 MAPK10 (0.45) MAPK10OPRK1PDE4DNR1I2ADORA3
Hydrochloric Acid SCHEMBL6718286 0.83 MAPK10 (0.53) MAPK10OPRK1PDE4DNR1I2ADORA3
Hydrochloric Acid SCHEMBL7402058 0.82 SRD5A2 (0.47) MAPK10OPRK1PDE4DNR1I2ADORA3
SCHEMBL6714765 0.81 CA1 (0.51) MAPK10OPRK1PDE4DNR1I2ADORA3
SCHEMBL2334077 0.81 MAPK10 (0.51) MAPK10MAPK9MAPK14ALDH1A1PLG
SCHEMBL28531265 0.81 MAPK10 (0.55) MAPK10OPRK1PDE4DNR1I2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110467548-B Sulfonamide or ketoamide compound and preparation method thereof 西南交通大学 2020-10-09 CN disclosed
CN-110467548-A A kind of sulfonamides or keto acyl aminated compounds and preparation method thereof UNIV SOUTHWEST JIAOTONG 2019-11-19 CN disclosed