SCHEMBL28341883

SCHEMBL28341883

C=CCN(CCc1ccccc1)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.43
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
BCHE P06276 3/20 0.40
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
GBA1 P04062 2/20 0.38
KCNA5 P22460 3/20 0.37
GPR52 Q9Y2T5 1/20 0.37
KCNN4 O15554 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
G6PC1 P35575 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28451780 0.85 TSHR (0.49) POLBMAPTMAPK1GAATSHR
SCHEMBL9763376 0.83 KCNA5 (0.39) POLBMAPTMAPK1KCNA5KCNN4
SCHEMBL12072374 0.77 CHRNB2 (0.41) POLBMAPTMAPK1TAAR1KCNA5
SCHEMBL28440491 0.77 KCNA5 (0.44) CHRNA7POLBMAPTMAPK1GAA
SCHEMBL9129445 0.74 CHRNA7 (0.57) CHRNA7GAATAAR1GBA1KCNA5
SCHEMBL18590700 0.73 TAAR1 (0.54) POLBMAPTMAPK1GAATSHR
SCHEMBL14415500 0.70 CHRNB2 (0.42) CHRNA7KCNA5KCNN4CYP2C19HDAC6
SCHEMBL11573309 0.69 OPRK1 (0.64) BCHETAAR1MEN1KMT2ASMN1; SMN2
SCHEMBL3749579 0.69 OPRK1 (0.59) BCHETAAR1MEN1KMT2ASMN1; SMN2
SCHEMBL18590701 0.68 GAA (0.53) POLBMAPTMAPK1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110627785-B Preparation method of 1, 5-tetrahydronaphthyridine derivative 温州大学 2021-06-25 CN disclosed
CN-110627785-A Preparation method of 1, 5-tetrahydronaphthyridine derivative 温州大学 2019-12-31 CN disclosed