SCHEMBL28344889

SCHEMBL28344889

C[Si](C)(C)C#Cc1ccc(O[SiH3])cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AR P10275 20/20 0.41
PGR P06401 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21839795 0.82 AR (0.40) ARPGR
SCHEMBL1914296 0.78 GABRA1 (0.36) ARPGR
SCHEMBL10088537 0.78 AR (0.45) AR
SCHEMBL30444423 0.76 AR (0.44) ARPGR
SCHEMBL1762439 0.76 GAA (0.47) ARPGR
SCHEMBL20535166 0.76 AR (0.44) ARPGR
SCHEMBL3347622 0.72 FFAR1 (0.40) AR
SCHEMBL17672783 0.71 NOTUM (0.52) AR
SCHEMBL1530568 0.69 CYP17A1 (0.48) AR
SCHEMBL20455567 0.68 PTGES (0.36) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678450-B Isoxazole derivatives as nuclear receptor agonists and uses thereof 日东制药株式会社 2023-06-20 CN disclosed
CN-110678450-A Isoxazole derivatives as nuclear receptor agonists and uses thereof 日东制药株式会社 2020-01-10 CN disclosed