SCHEMBL3347622

SCHEMBL3347622

C[Si](C)(C)C#Cc1ccccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HSD11B1 P28845 4/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
NOTUM Q6P988 2/20 0.35
PTGES O14684 3/20 0.33
AR P10275 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8960256 0.82 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1CYP1A2CYP3A4
SCHEMBL17940722 0.82 KDM4E (0.36) ALDH1A1KDM4EMEN1CYP1A2CYP3A4
SCHEMBL7677291 0.82 MRGPRX1 (0.39) ALDH1A1KDM4EMEN1CYP1A2CYP3A4
SCHEMBL27896461 0.80 SLC22A12 (0.35) ALDH1A1KDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL3839029 0.79 KDM4E (0.49) ALDH1A1KDM4EMEN1CYP1A2CYP3A4
SCHEMBL5250349 0.78 FFAR1 (0.43) FFAR1ALDH1A1MEN1CYP1A2MAPT
SCHEMBL10088537 0.77 AR (0.45) AR
SCHEMBL1914296 0.77 GABRA1 (0.36) AR
SCHEMBL20455567 0.77 PTGES (0.36) HSD11B1PTGESAR
SCHEMBL20535166 0.75 AR (0.44) ALDH1A1CYP2C9HSD17B10AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055947-A1 ALKYNE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-04-14 WO disclosed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed