SCHEMBL28344922

SCHEMBL28344922

C[Si](C)(C)CCc1ccc(O[SiH3])cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.36
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
MAOB P27338 2/20 0.33
CALM1 P0DP23 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PPARA Q07869 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
AOC3 Q16853 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
F2RL1 P55085 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28881522 0.89 MAOB (0.31) TAAR1ALDH1A1POLBMAOB
SCHEMBL15952484 0.82 ESR1 (0.40) TAAR1HRH3KDM4ELMNA
SCHEMBL28906287 0.76 SMN1; SMN2 (0.35) TAAR1ALDH1A1POLBSMN1; SMN2PPARA
SCHEMBL28906297 0.75 DAO (0.34) TAAR1ALDH1A1POLBSMN1; SMN2PPARA
SCHEMBL24602755 0.73 CYP1A2 (0.52) TAAR1ALDH1A1SMN1; SMN2HRH3
SCHEMBL17722492 0.73 LPL (0.46) ALDH1A1
SCHEMBL20536283 0.72 PPARA (0.35) TAAR1ALDH1A1POLBCALM1PPARA
SCHEMBL3211356 0.71 GFER (0.59) TAAR1ALDH1A1MAOBSMN1; SMN2
SCHEMBL21925685 0.71 CA2 (0.41) PPARA
SCHEMBL20004512 0.71 TAAR1 (0.50) TAAR1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678450-B Isoxazole derivatives as nuclear receptor agonists and uses thereof 日东制药株式会社 2023-06-20 CN disclosed
CN-110678450-A Isoxazole derivatives as nuclear receptor agonists and uses thereof 日东制药株式会社 2020-01-10 CN disclosed