SCHEMBL28345416

SCHEMBL28345416

Cc1coc(-c2ccnc(NC(C)(C)C)n2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
CDC7 O00311 1/20 0.34
MAP4K4 O95819 1/20 0.34
PIM1 P11309 1/20 0.34
PRKACA P17612 1/20 0.34
GSK3B P49841 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
SRC P12931 7/20 0.34
SYK P43405 7/20 0.34
ZAP70 P43403 6/20 0.34
CDK2 P24941 3/20 0.33
NPC1 O15118 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30209592 1.00 PIK3CD (0.36) PIK3CDPIK3C3MAPK13MAPK12MAPK11
SCHEMBL28343115 0.74 PIK3CD (0.37) PIK3CDPIK3C3MAPK13MAPK12MAPK11
SCHEMBL28345339 0.72 CDK4 (0.30)
SCHEMBL28342721 0.72 LMNA (0.44) MAPK13MAPK12MAPK11MAPK14CDK2
SCHEMBL30209582 0.72 LMNA (0.44) MAPK13MAPK12MAPK11MAPK14CDK2
SCHEMBL28345474 0.70 KDM4E (0.39) NPC1RAB9AKDM4EALDH1A1GLA
SCHEMBL30209584 0.70 KDM4E (0.39) NPC1RAB9AKDM4EALDH1A1GLA
SCHEMBL12410773 0.69 NPSR1 (0.45) NPC1RAB9AALDH1A1
SCHEMBL23244457 0.67 PLK1 (0.43) MAPK13PIM1GSK3BSYKCDK2
SCHEMBL3653788 0.67 DKK1 (0.52) MAPK13MAPK12MAPK11MAPK14CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110655509-B 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-01-24 CN disclosed
CN-110684020-B 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-01-20 CN disclosed
CN-110684020-A 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-01-14 CN disclosed
CN-110655509-A 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-01-07 CN disclosed