SCHEMBL28345474

SCHEMBL28345474

Cc1coc(-c2ccnc(S(C)(=O)=O)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 5/20 0.39
RAB9A P51151 4/20 0.39
TP53 P04637 3/20 0.39
STAT3 P40763 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 2/20 0.39
HSD17B10 Q99714 2/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
JAK2 O60674 1/20 0.39
TLR8 Q9NR97 1/20 0.39
SDHB P21912 4/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 3/20 0.36
BPTF Q12830 2/20 0.33
DYRK1A Q13627 1/20 0.33
DYRK2 Q92630 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30209584 1.00 KDM4E (0.39) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL21621272 0.77 ALDH1A1 (0.58) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL30107948 0.77 ALDH1A1 (0.58) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL28822645 0.73 KDM4E (0.35) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL30209582 0.73 LMNA (0.44) KDM4EALDH1A1NPSR1HPGDHTT
SCHEMBL28342721 0.73 LMNA (0.44) KDM4EALDH1A1NPSR1HPGDHTT
SCHEMBL4138614 0.71 NPSR1 (0.42) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL30637352 0.71 NPSR1 (0.42) KDM4EALDH1A1RAB9ATP53STAT3
SCHEMBL2199521 0.71 GRM4 (0.59) KDM4EALDH1A1RAB9ATP53HPGD
SCHEMBL3580841 0.71 MAP4K4 (0.43) KDM4EALDH1A1RAB9ATP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110655509-B 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-01-24 CN disclosed
CN-110684020-A 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-01-14 CN disclosed
CN-110655509-A 2-aminopyrimidine derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-01-07 CN disclosed