SCHEMBL28347478

SCHEMBL28347478

Cc1c(F)cccc1OC(=O)N1CCC(C(CCCOCc2ccccc2)NC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.42
PPARG P37231 2/20 0.38
CCR1 P32246 1/20 0.37
CHRM2 P08172 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CASP3 P42574 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
SLC6A12 P48065 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
MCHR1 Q99705 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22023439 1.00 CCKBR (0.42) CCKBRPPARGCCR1CHRM2MAPT
SCHEMBL20601122 0.90 NPSR1 (0.38) CCR1CHRM2MAPTTSHRCASP3
SCHEMBL20601121 0.90 NPSR1 (0.38) CCR1CHRM2MAPTTSHRCASP3
SCHEMBL20600893 0.88 PLD2 (0.38) CCR1CHRM2MAPTTSHRCASP3
SCHEMBL20600894 0.88 PLD2 (0.38) CCR1CHRM2MAPTTSHRCASP3
SCHEMBL20600981 0.85 CCKBR (0.43) CCKBRCCR1MEN1KMT2ASLC6A12
SCHEMBL20600979 0.85 CCKBR (0.43) CCKBRCCR1MEN1KMT2ASLC6A12
SCHEMBL20615629 0.85 GPR119 (0.47) MEN1KMT2AL3MBTL1LMNA
SCHEMBL28347947 0.85 GPR119 (0.47) MEN1KMT2AL3MBTL1LMNA
SCHEMBL20601115 0.83 PLD2 (0.41) CCR1CHRM2MAPTTSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110709391-A Modulators of indoleamine2, 3-dioxygenase 葛兰素史克知识产权开发有限公司 2020-01-17 CN disclosed