SCHEMBL28348449

SCHEMBL28348449

CCOC(=O)c1cccc(F)c1NC(=O)c1cn(C)nc1C(F)F

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.48
MAPT P10636 1/20 0.47
KDM4E B2RXH2 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NLRP3 Q96P20 1/20 0.40
POLB P06746 1/20 0.40
JMJD6 Q6NYC1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
BTK Q06187 1/20 0.40
DHODH Q02127 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28345018 0.88 LMNA (0.51) LMNAMAPTKDM4ESMN1; SMN2NPC1
SCHEMBL28348535 0.88 TP53 (0.42) LMNAMAPTKDM4ESMN1; SMN2NPC1
SCHEMBL28350646 0.85 KMT2A (0.43) KDM4ETDP1POLBL3MBTL1DHODH
SCHEMBL28345856 0.84 LMNA (0.51) LMNAMAPTKDM4ESMN1; SMN2NPC1
SCHEMBL973238 0.81 ATM (0.47) DHODH
SCHEMBL972255 0.81 EGFR (0.48) SMN1; SMN2DHODH
SCHEMBL22029397 0.81 POLB (0.47) MAPTKDM4ESMN1; SMN2NPC1ALDH1A1
SCHEMBL19186 0.80 JMJD6 (0.44) LMNAKDM4ENPC1RAB9AALDH1A1
SCHEMBL3685890 0.78 HTT (0.43) LMNAKDM4ERAB9ATP53HTT
SCHEMBL28348547 0.78 NPSR1 (0.42) LMNAMAPTKDM4ESMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110615765-B (1H-pyrazole-4-formamido) ethyl benzoate compound and preparation method and application thereof 浙江工业大学 2021-06-25 CN disclosed
CN-110615765-A (1H-pyrazole-4-formamido) ethyl benzoate compound and preparation method and application thereof 浙江工业大学 2019-12-27 CN disclosed