SCHEMBL28352964

SCHEMBL28352964

Cc1cc2c(CCc3ccc(C(F)(F)F)cc3)ccc(C#N)c2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DAO P14920 6/20 0.43
MRGPRX4 Q96LA9 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
AR P10275 4/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
MAPT P10636 1/20 0.33
OPRL1 P41146 1/20 0.33
HRH1 P35367 1/20 0.33
HTR6 P50406 1/20 0.33
MIF P14174 1/20 0.33
NR1H2 P55055 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28356899 0.81 DAO (0.45) DAOTAAR1MAPTOPRL1
SCHEMBL29259245 0.75 AR (0.43) ARMAPT
SCHEMBL29259242 0.75 DHODH (0.43)
SCHEMBL28352950 0.75 AR (0.43) ARMAPT
SCHEMBL28356859 0.74 NQO2 (0.39) ARMAPT
SCHEMBL29259243 0.73 TOP2A (0.37) ARMAPT
SCHEMBL28958657 0.71 PARP1 (0.42) MAPT
SCHEMBL21008875 0.70 TRPV4 (0.39) ARPDE3BPDE3A
SCHEMBL28882601 0.70 AR (0.43) AR
SCHEMBL22439122 0.68 DAO (0.38) DAOMRGPRX4TAAR1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110770211-B Alpha, beta unsaturated amide compound 协和麒麟株式会社 2023-09-19 CN disclosed
CN-110770211-A α unsaturated amide compound 协和麒麟株式会社 2020-02-07 CN disclosed