SCHEMBL28354444

SCHEMBL28354444

COc1cccc(C2(N)CC(=O)c3ccccc3O2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIB P23284 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP19A1 P11511 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KLK7 P49862 1/20 0.42
MAPT P10636 3/20 0.41
HPGD P15428 1/20 0.41
KDM1A O60341 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
UTS2R Q9UKP6 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7118017 0.82 PPIB (0.43) PPIBALDH1A1KDM4ECYP19A1SMN1; SMN2
SCHEMBL927371 0.81 SIGMAR1 (0.45) ALDH1A1KDM4ECYP19A1SMN1; SMN2MAPT
SCHEMBL27288753 0.81 SIGMAR1 (0.45) ALDH1A1KDM4ECYP19A1SMN1; SMN2MAPT
SCHEMBL11013389 0.70 MEN1 (0.43) ALDH1A1KDM1ASIGMAR1MEN1KMT2A
SCHEMBL30872986 0.70 RIPK1 (0.53) PPIBALDH1A1KDM4ECYP19A1SMN1; SMN2
SCHEMBL7154660 0.70 MAOB (0.47) PPIBALDH1A1KDM4ECYP19A1SMN1; SMN2
SCHEMBL29757571 0.69 MAOB (0.39) ALDH1A1KDM4ESMN1; SMN2MAPTHPGD
SCHEMBL6191270 0.69 ALDH1A1 (0.43) PPIBALDH1A1KDM4ECYP19A1SMN1; SMN2
SCHEMBL2120395 0.69 ATM (0.44) PPIBKDM4ECYP19A1SMN1; SMN2MAPT
SCHEMBL29375243 0.68 KDM4E (0.60) PPIBALDH1A1KDM4ECYP19A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113329792-B Substituted 3- (1-oxo-isoindolin-2-yl) piperidine-2, 6-dione derivatives and uses thereof 诺华股份有限公司 2024-06-28 CN disclosed
CN-112585136-B Urea compounds and compositions as SMARCA2/BRM atpase inhibitors 诺华股份有限公司 2024-06-25 CN disclosed
CN-117794929-A Selective BCL-XL PROTAC compounds and methods of use 法国施维雅药厂 2024-03-29 CN disclosed
CN-117500803-A Amino-substituted heterocycles for the treatment of cancers with EGFR mutations 纽威伦特公司 2024-02-02 CN disclosed
CN-117355333-A Combination comprising anti-TM 4SF1 antibody and immunotherapeutic agent and method of use thereof 安吉克公司 2024-01-05 CN disclosed
CN-117355304-A ALK-5 inhibitors and uses thereof 住友制药肿瘤公司 2024-01-05 CN disclosed
CN-117122707-A combination therapy 意大利国际先进加速器应用有限公司 2023-11-28 CN disclosed
CN-117098776-A Use of anti-TGF-beta antibodies and other therapeutic agents for the treatment of proliferative diseases 诺华股份有限公司 2023-11-21 CN disclosed
CN-116829143-A Forms and formulations of non-receptor tyrosine kinase 1 (TNK 1) inhibitors 住友制药肿瘤公司 2023-09-29 CN disclosed
CN-116761635-A BCL-XL inhibitor antibody drug conjugates and methods of use thereof 诺华股份有限公司 2023-09-15 CN disclosed
CN-112867512-A Combination therapy 意大利国际先进加速器应用有限公司 2021-05-28 CN disclosed
CN-112585136-A Urea compounds and compositions as SMARCA2/BRM ATPase inhibitors 诺华股份有限公司 2021-03-30 CN disclosed
CN-112584875-A Stabilized, concentrated solutions of radionuclide complexes 先进加速器应用公司 2021-03-30 CN disclosed
CN-112334194-A 3- (5-amino-1-oxoisoindolin-2-yl) piperidine-2, 6-dione derivatives and their use in the treatment of IKAROS family Zinc finger 2(IKZF2) dependent diseases 诺华股份有限公司 2021-02-05 CN disclosed
CN-112261970-A 3- (5-hydroxy-1-oxoisoindolin-2-yl) piperidine-2, 6-dione derivatives and their use in the treatment of IKAROS family Zinc finger 2(IKZF2) dependent diseases 诺华股份有限公司 2021-01-22 CN disclosed
CN-111107868-A Antibody cytokine transplantation proteins and methods of use 诺华股份有限公司 2020-05-05 CN disclosed
CN-111032085-A Combination of an immune checkpoint antagonist and a RANK-L (NF-KB ligand) antagonist or bispecific binding molecules thereof for use in cancer treatment or prevention and uses thereof 昆士兰医学研究所理事会 2020-04-17 CN disclosed
CN-110799218-A Antibody conjugates comprising STING agonists 诺华股份有限公司 2020-02-14 CN disclosed
CN-110678183-A Antibody conjugates comprising TOLL-like receptor agonists and combination therapies 诺华股份有限公司 2020-01-10 CN disclosed
CN-110662762-A Antibody cytokine transplantation proteins and methods for treating cancer 诺华股份有限公司 2020-01-07 CN disclosed