SCHEMBL28356916

SCHEMBL28356916

O=C(C=Cc1ccc(O)cc1)C=Cc1cccnc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.81
RAB9A P51151 2/20 0.81
KDM4E B2RXH2 2/20 0.81
JUN P05412 2/20 0.81
NFKB1 P19838 2/20 0.81
NPC1 O15118 1/20 0.81
MAPK1 P28482 1/20 0.81
GPR55 Q9Y2T6 1/20 0.81
KMT2A Q03164 1/20 0.70
CYP2D6 P10635 6/20 0.65
CYP2C9 P11712 2/20 0.65
F3 P13726 2/20 0.65
TYR P14679 1/20 0.65
HSD11B1 P28845 1/20 0.65
USP2 O75604 1/20 0.57
PFKFB3 Q16875 1/20 0.56
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
CYP1A2 P05177 8/20 0.53
CYP1A1 P04798 7/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5598852 0.90 MAPT (1.00) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL5598850 0.90 MAPT (1.00) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL16093039 0.88 MAPT (0.89) MAPTRAB9AKDM4EJUNNFKB1
Hydrochloric Acid SCHEMBL11971085 0.88 MAPT (0.96) MAPTRAB9AKDM4EJUNNFKB1
Hydrochloric Acid SCHEMBL11971079 0.88 MAPT (0.96) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL11067983 0.86 CYP11B1 (0.70) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL9605429 0.86 CYP11B1 (0.70) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL11067984 0.86 CYP11B1 (0.70) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL1604140 0.83 RAB9A (1.00) MAPTRAB9AKDM4EJUNNFKB1
SCHEMBL29600034 0.83 RAB9A (1.00) MAPTRAB9AKDM4EJUNNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530435-B Quinoxaline-containing 1, 4-pentadiene-3-ketone derivative, preparation method and application 贵州大学 2021-08-17 CN disclosed
CN-106928176-B Coumarin-containing 1, 4-pentadiene-3-ketone derivative and preparation method and application thereof 贵州大学 2020-02-18 CN disclosed