SCHEMBL2835830

SCHEMBL2835830

Cc1nc(-c2ncccc2OCc2ccccc2)n(CCc2ccccc2)c(=O)c1-c1cc(-c2ccccn2)c(C)s1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASR P41180 13/20 0.66
NR1I2 O75469 5/20 0.52
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
TSHR P16473 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 1/20 0.38
HIF1A Q16665 1/20 0.38
MCL1 Q07820 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GRM5 P41594 1/20 0.34
BRD4 O60885 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2843300 0.88 CASR (0.52) CASRNR1I2GRM5
SCHEMBL2837296 0.87 CASR (0.49) CASRNR1I2ALDH1A1CYP1A2CYP3A4
SCHEMBL2840722 0.87 CASR (0.73) CASRNR1I2
Hydrochloric Acid SCHEMBL2835851 0.87 CASR (0.72) CASRNR1I2
SCHEMBL2838847 0.84 CASR (0.55) CASRNR1I2ALDH1A1CYP1A2CYP3A4
SCHEMBL3345007 0.83 CASR (0.80) CASRNR1I2ALDH1A1CYP1A2CYP3A4
SCHEMBL13418278 0.80 CASR (0.86) CASRNR1I2
SCHEMBL4147810 0.80 CASR (0.56) CASRNR1I2ALDH1A1CYP1A2CYP3A4
SCHEMBL3344554 0.79 CASR (1.00) CASRNR1I2
Hydrochloric Acid SCHEMBL3345010 0.79 CASR (0.98) CASRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed