SCHEMBL2837296

SCHEMBL2837296

Cc1nc(-c2ncccc2OCc2ccccc2)n(CCc2ccccc2)c(=O)c1-c1cc(Br)c(C)s1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.49
NR1I2 O75469 4/20 0.44
ALDH1A1 P00352 5/20 0.40
CYP1A2 P05177 4/20 0.40
TSHR P16473 4/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2C19 P33261 3/20 0.40
LMNA P02545 1/20 0.40
HIF1A Q16665 1/20 0.40
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK14 Q16539 1/20 0.35
USP2 O75604 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GCK P35557 1/20 0.34
CYP2D6 P10635 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2835830 0.87 CASR (0.66) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2838847 0.87 CASR (0.55) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2839722 0.83 TSHR (0.46) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL4147810 0.80 CASR (0.56) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL3345000 0.80 CASR (0.60) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2858671 0.78 BRD4 (0.43) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL4144136 0.78 CASR (0.51) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2839694 0.77 CYP1A2 (0.43) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2843300 0.76 CASR (0.52) CASRNR1I2
SCHEMBL2838115 0.76 CASR (0.55) CASRALDH1A1CYP1A2TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed