SCHEMBL2838847

SCHEMBL2838847

Cc1ccc(-c2c(C)nc(-c3ncccc3OCc3ccccc3)n(CCc3ccccc3)c2=O)s1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.55
NR1I2 O75469 4/20 0.55
ALDH1A1 P00352 4/20 0.43
CYP1A2 P05177 4/20 0.43
TSHR P16473 4/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP3A4 P08684 3/20 0.43
LMNA P02545 1/20 0.43
HIF1A Q16665 1/20 0.43
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PIK3C2A O00443 1/20 0.37
USP2 O75604 2/20 0.37
GCK P35557 1/20 0.36
CYP2D6 P10635 1/20 0.36
GFER P55789 1/20 0.36
LTA4H P09960 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138510 0.88 CASR (0.67) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2837296 0.87 CASR (0.49) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2839040 0.85 CASR (0.63) CASRNR1I2PIK3C2A
SCHEMBL2835830 0.84 CASR (0.66) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2839722 0.83 TSHR (0.46) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2839694 0.80 CYP1A2 (0.43) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL2858671 0.80 BRD4 (0.43) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL4142850 0.79 NR1I2 (0.70) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL4142963 0.79 CASR (0.57) CASRNR1I2ALDH1A1CYP1A2TSHR
SCHEMBL4143278 0.78 CASR (0.54) CASRNR1I2ALDH1A1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed