SCHEMBL28360378

SCHEMBL28360378

COC(=O)C(C)N=Cc1ccco1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.49
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
POLB P06746 5/20 0.45
TDP1 Q9NUW8 3/20 0.45
CTDSP1 Q9GZU7 2/20 0.44
AHR P35869 1/20 0.44
PLA2G7 Q13093 1/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28465909 0.85 MAPT (0.46) MAPTALDH1A1KDM4EHPGDMAPK1
SCHEMBL11651918 0.75 ALDH1A1 (0.63) MAPTALDH1A1KDM4EHPGDMAPK1
SCHEMBL11651924 0.75 ALDH1A1 (0.63) MAPTALDH1A1KDM4EHPGDMAPK1
SCHEMBL5303065 0.74 MAPT (0.49) MAPTALDH1A1KDM4EPOLBTDP1
SCHEMBL5303064 0.74 MAPT (0.49) MAPTALDH1A1KDM4EPOLBTDP1
SCHEMBL1962034 0.74 MIF (0.52) PLA2G7NPC1RAB9ASMN1; SMN2GAA
SCHEMBL8259717 0.74 MIF (0.52) PLA2G7NPC1RAB9ASMN1; SMN2GAA
SCHEMBL13201409 0.74 MIF (0.52) PLA2G7NPC1RAB9ASMN1; SMN2GAA
SCHEMBL8126152 0.74 MIF (0.52) PLA2G7NPC1RAB9ASMN1; SMN2GAA
SCHEMBL1962036 0.74 MIF (0.52) PLA2G7NPC1RAB9ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110669046-B Polysubstituted tetrahydro-gamma-carboline derivative with multiple chiral centers and preparation method of stereo diversity of polysubstituted tetrahydro-gamma-carboline derivative 武汉大学 2021-07-06 CN disclosed
CN-110669046-A Polysubstituted tetrahydro-gamma-carboline derivative with multiple chiral centers and preparation method of stereo diversity of polysubstituted tetrahydro-gamma-carboline derivative 武汉大学 2020-01-10 CN disclosed